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Parsaclisib hydrochloride
Parsaclisib hydrochloride (INCB050465 HCl) is a selectve PI3Kδ inhibitor with antitumor activity. Parsaclisib demonstrates potent activity with IC50 values ranging from 0.2 to 2 nM.
Catalog No. T28297Cas No. 1995889-48-9
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Parsaclisib hydrochloride
Catalog No. T28297Alias Parsaclisib HCl, INCB-50465, INCB 050465, INCB-050465, INCB050465 HCl, INCB 50465, INCB50465 HClCas No. 1995889-48-9
Parsaclisib hydrochloride (INCB050465 HCl) is a selectve PI3Kδ inhibitor with antitumor activity. Parsaclisib demonstrates potent activity with IC50 values ranging from 0.2 to 2 nM.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,230 | 1-2 weeks | |
| 50 mg | $1,610 | 1-2 weeks | |
| 100 mg | $2,570 | 1-2 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Parsaclisib hydrochloride (INCB050465 HCl) is a selectve PI3Kδ inhibitor with antitumor activity. Parsaclisib demonstrates potent activity with IC50 values ranging from 0.2 to 2 nM. |
| Targets&IC50 | PI3Kδ:1 nM (IC50) |
| Alias | Parsaclisib HCl, INCB-50465, INCB 050465, INCB-050465, INCB050465 HCl, INCB 50465, INCB50465 HCl |
| Molecular Weight | 469.34 |
| Formula | C20H23Cl2FN6O2 |
| Cas No. | 1995889-48-9 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 90 mg/mL (191.76 mM) H2O: Insoluble | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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